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approved_drugs

Track hit to lead campaigns of all approved small molecules

Alt text

List

2019

  • alpelisib (Piqray; Novartis)
  • erdafitinib (Balversa; Astex -> Janssen)
  • darolutamide (Nubeqa; Orion -> Bayer)
  • fedratinib (Inrebic; TargeGen -> Sanofi -> Celgene)
  • selinexor (Xpovio; Karyopharm Therapeutics)
  • entrectinib (Rozlytrek; Roche)

2018

  • glasdegib (Daurismo; Pfizer)